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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T16369 | O-Desmethyl gefitinib | EGFR | |
O-Desmethyl gefitinib inhibits EGFR (IC50: 36 nM in subcellular assays). In human plasma, O-Desmethyl gefitinib is an active metabolite of Gefitinib. The formation of O-desmethyl gefitinib is dependent on the CYP2D6 acti... | |||
T19489 | O-Desmethyl gefitinib D8 | EGFR | |
O-Desmethyl gefitinib D8 is a deuterium labeled O-Desmethyl gefitinib that is an active metabolite of Gefitinib in human plasma. |